Opaganib-[13C6]
Opaganib-[13C6] is the labelled analogue of Opaganib. Opaganib is an orally available, aryladamantane compound and selective inhibitor of sphingosine kinase-2 (SK2) with potential antineoplastic activity. Upon administration, Opaganib competitively binds to and inhibits SK2, thereby preventing the phosphorylation of the pro-apoptotic amino alcohol sphingosine to sphingosine 1-phosphate (S1P), the lipid mediator that is pro-survival and critical for immunomodulation.
Supplier | BOC Sciences |
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Product # | BLP-000773 |
Pricing | Inquire |
Molecular Weight | 386.87 |
Molecular Formula | C17[13C]6H25ClN2O |