GRK2-IN-1 hydrochloride

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Supplier MedChemExpress
Product # HY-109562A-5 mg
Pricing 5 mg, USD $350.0
Biological Activity
  • GRKs-IN-1 hydrochloride, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=130 nM) and GRK5 (IC50=7.1 μM).
  • GRKs-IN-1 hydrochloride is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine[1].
Purity 98.23%
MWt 488.94
Formula C₂₄H₂₆ClFN₄O₄
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