Facinicline hydrochloride
Supplier | MedChemExpress |
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Product # | HY-108057A-5 mg |
CAS # | 677305-02-1 |
Pricing | 5 mg, USD $300.0 |
Synonyms | RG3487 hydrochloride |
MWt | 306.79 |
Formula | C₁₅H₁₉ClN₄O |
Biological Activity | Facinicline hydrochloride (RG3487 hydrochloride) is an orally active nicotinic α7 receptor partial agonist, with a Ki of 6 nM for α7 human nAChR. Facinicline hydrochloride (RG3487 hydrochloride) improves cognition and sensorimotor gating in rodents. Facinicline hydrochloride (RG3487 hydrochloride) shows high affinity (antagonist) to 5-HT3Rs with a Ki value of 1.2 nM[1]. |
Purity | 99.93% |