Asimadoline
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-107384-10 mM * 1 mL |
| CAS # | 153205-46-0 |
| Pricing | 10 mM * 1 mL, USD $92.0 |
| Synonyms | EMD-61753 |
| MWt | 414.54 |
| Formula | C₂₇H₃₀N₂O₂ |
| Biological Activity | Asimadoline (EMD-61753) is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline has low permeability across the blood brain barrier and has peripheral anti-inflammatory actions. Asimadoline ameliorates allodynia in diabetic rats and has the potential for irritable bowel syndrome (IBS)[1][2][3]. |
| Purity | 99.36% |