Prinaberel
Supplier | MedChemExpress |
---|---|
Product # | HY-14933-50 mg |
CAS # | 524684-52-4 |
Pricing | 50 mg, USD $648.0 |
Synonyms | ERB-041 |
MWt | 271.24 |
Formula | C₁₅H₁₀FNO₃ |
Biological Activity | Prinaberel (ERB-041) is a potent and selective estrogen receptor (ER) β agonist with IC50s of 5.4, 3.1 and 3.7 nM for human, rat and mouse ERβ, respectively. Prinaberel displays >200-fold selectivity for ERβ over ERα. Prinaberel is a potent skin cancer chemopreventive agent that acts by dampening the WNT/β-catenin signaling pathway. Prinaberel induces ovarian cancer apoptosis[1][2][3]. |
Purity | 98.62% |