CALP1 TFA
Supplier | MedChemExpress |
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Product # | HY-P1077A |
Pricing | inquire |
Biological Activity | CALP1 TFA is a calmodulin (CaM) agonist (Kd of 88 µM) with binding to the CaM EF-hand/Ca2+-binding site. CALP1 TFA blocks calcium influx and apoptosis (IC50 of 44.78 µM) through inhibition of calcium channel opening. CALP1 TFA blocks glutamate receptor channels and blocks a store-operated nonselective cation channel. CALP1 TFA activates CaM-dependent phosphodiesterase activity[1][2][3][4]. |
MWt | 956.1 |
Formula | C₄₂H₇₆F₃N₉O₁₂ |