Birabresib (OTX015)

Birabresib (OTX015, MK 8628) is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4 in cell-free assays. Birabresib inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.
Supplier Selleck Chemicals
Product # S7360
Sku # S7360-10mM/1mL
Pricing 10mM/1mL, $197.00
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