Birabresib (OTX015)
![](https://image.labshake.com/supplier-product/471d3a2a-073f-4b25-a7de-2da1c79248d6/254e84f8-f2b4-4875-937b-fa99cbd8adec.png)
Birabresib (OTX015, MK 8628) is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4 in cell-free assays. Birabresib inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.
Supplier | Selleck Chemicals |
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Product # | S7360 |
Sku # | S7360-10mM/1mL |
Pricing | 10mM/1mL, $197.00 |