HET0016
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-124527-100 mg |
| CAS # | 339068-25-6 |
| Pricing | 100 mg, USD $650.0 |
| Biological Activity | HET0016 is a potent and selective 20-hydroxyeicosatetraenoic acid (20-HETE) synthase inhibitor, with IC50 values of 17.7 nM, 12.1 nM and 20.6 nM for recombinant CYP4A1-, CYP4A2- and CYP4A3-catalyzed 20-HETE synthesis, respectively. HET0016 also is a selective CYP450 inhibitor, which has been shown to inhibit angiogenesis and tumor growth[1][2]. |
| Purity | 99.78% |
| MWt | 206.28 |
| Formula | C₁₂H₁₈N₂O |