Acolbifene
Supplier | MedChemExpress |
---|---|
Product # | HY-16023A-10 mg |
CAS # | 182167-02-8 |
Pricing | 10 mg, USD $350.0 |
Synonyms | EM-652; SCH 57068 |
MWt | 457.56 |
Formula | C₂₉H₃₁NO₄ |
Biological Activity | Acolbifene (EM-652), the active metabolite of EM800, is an orally active pure antiestrogen and selective estrogen receptor antagonist. Acolbifene (EM-652) inhibits estradiol (E2)-induced transcriptional activity of ERα (IC50 = 2 nM) and ERβ (IC50 = 0.4 nM). Acolbifene (EM-652) possesses potent and pure anticarcinogenic properties[1][2][3][4][5]. |
Purity | 98.86% |