Timapiprant sodium
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-15342A-10 mM * 1 mL |
| CAS # | 950688-14-9 |
| Pricing | 10 mM * 1 mL, USD $77.0 |
| Synonyms | OC000459 sodium |
| MWt | 370.35 |
| Formula | C₂₁H₁₆FN₂NaO₂ |
| Biological Activity | Timapiprant sodium (OC000459 sodium) is a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist. Timapiprant sodium (OC000459 sodium) potently displaces [3H] PGD2 from human recombinant DP2 (Ki=13 nM), rat recombinant DP2 (Ki=3 nM), and human native DP2 (Ki=4 nM). Timapiprant sodium (OC000459 sodium) inhibits mast cell activation of Th2 lymphocytes and eosinophils[1]. |
| Purity | ≥98.0% |