Timapiprant sodium

Supplier MedChemExpress
Product # HY-15342A-10 mM * 1 mL
CAS # 950688-14-9
Pricing 10 mM * 1 mL, USD $77.0
Synonyms OC000459 sodium
MWt 370.35
Formula C₂₁H₁₆FN₂NaO₂
Biological Activity Timapiprant sodium (OC000459 sodium) is a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist. Timapiprant sodium (OC000459 sodium) potently displaces [3H] PGD2 from human recombinant DP2 (Ki=13 nM), rat recombinant DP2 (Ki=3 nM), and human native DP2 (Ki=4 nM). Timapiprant sodium (OC000459 sodium) inhibits mast cell activation of Th2 lymphocytes and eosinophils[1].
Purity ≥98.0%
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