Antihistamine-1
Antihistamine-1 is an H1-antihistamine (Ki = 6.9 nM) with acceptable blood-brain barrier penetration. It is also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
| Supplier | BOC Sciences |
|---|---|
| Product # | 1186430-60-3 |
| Pricing | Inquire |
| Cas | 1186430-60-3 |
| Molecular Weight | 389.47 |
| Molecular Formula | C23H24FN5 |
| Canonical SMILES | CC1=CN(N=C1)C2CCN(CC2)C3=NC4=CC=CC=C4N3CC5=CC=C(C=C5)F |