GDC-0276
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-114237-5 mg |
| CAS # | 1494581-70-2 |
| Pricing | 5 mg, USD $450.0 |
| Biological Activity | GDC-0276 is a potent, selective, reversible and orally active NaV1.7 inhibitor with an IC50 value of 0.4 nM. GDC-0276 is well tolerated and exhibits a good pharmacokinetic profile. GDC-0276 has the potential for the treatment of pain and to address shortcomings of existing pain medications, such as addiction and off-target side effects[1]. |
| Purity | 99.51% |
| MWt | 462.58 |
| Formula | C₂₄H₃₁FN₂O₄S |