ML221
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-103254-50 mg |
| CAS # | 877636-42-5 |
| Pricing | 50 mg, USD $390.0 |
| Biological Activity | ML221 is a potent apelin (APJ) functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays. |
| Purity | ≥98.0% |
| MWt | 385.35 |
| Formula | C₁₇H₁₁N₃O₆S |