CGP 12177
CGP 12177 is a partial β3-adrenoceptor agonist with Ki value of 88 nM. It is also an of β1- and β2-adrenoceptors antagonist with Ki values of 0.9 nM and 4 nM for β1-, β2adrenoceptors. CGP12177 can slightly activate L-type Ca2+ current in human ventricular myocytes.
| Supplier | BOC Sciences |
|---|---|
| Product # | 81047-99-6 |
| Pricing | Inquire |
| Cas | 81047-99-6 |
| Molecular Weight | 279.34 |
| Molecular Formula | C14H21N3O3 |
| Canonical SMILES | CC(C)(C)NCC(COc1cccc2c1[nH]c(=O)[nH]2)O |