CK2/ERK8-IN-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-135906-10 mM * 1 mL |
| CAS # | 1085822-09-8 |
| Pricing | 10 mM * 1 mL, USD $88.0 |
| Biological Activity | CK2/ERK8-IN-1 is a dual casein kinase 2 (CK2) (Ki of 0.25 µM) and ERK8 (MAPK15, ERK7) inhibitor with IC50s of 0.50 μM. CK2/ERK8-IN-1 also binds to PIM1, HIPK2 (homeodomain-interacting protein kinase 2), and DYRK1A with Kis of 8.65 µM, 15.25 µM, and 11.9 µM, respectively. CK2/ERK8-IN-1 has pro-apoptotic efficacy[1]. |
| Purity | ≥99.0% |
| MWt | 534.82 |
| Formula | C₁₁H₉Br₄N₃O₂ |