BMX-IN-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-80002-50 mg |
| CAS # | 1431525-23-3 |
| Pricing | 50 mg, USD $750.0 |
| Synonyms | BMX kinase inhibitor |
| MWt | 524.59 |
| Formula | C₂₉H₂₄N₄O₄S |
| Biological Activity | BMX-IN-1 is a selective, irreversible inhibitor of bone marrow tyrosine kinase on chromosome X (BMX) that targets Cys496 in the BMX ATP binding domain with an IC50 of 8 nM, also targets the related Bruton’s tyrosine kinase (BTK) with an IC50 value of 10.4 nM, but is more than 47-656-fold less potent against Blk, JAK3, EGFR, Itk, or Tec activity. |
| Purity | 99.04% |