GSK484 hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-100514-10 mM * 1 mL |
| CAS # | 1652591-81-5 |
| Pricing | 10 mM * 1 mL, USD $213.0 |
| Biological Activity | GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 (PAD4) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed. |
| MWt | 510.03 |
| Formula | C₂₇H₃₂ClN₅O₃ |