WDR5-IN-4 TFA

Supplier MedChemExpress
Product # HY-111753A-10 mg
Pricing 10 mg, USD $550.0
Biological Activity WDR5-IN-4 TFA is an inhibitor of the WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5), with a Kd of 0.1 nM. WDR5-IN-4 TFA displaces WDR5 from chromatin and decreases the expression of associated genes, causing translational inhibition, nucleolar stress. Anti-cancer activity[1].
Purity 98.43%
MWt 612.4
Formula C₂₇H₂₃Cl₂F₄N₅O₃
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