CPI-455
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-100421-50 mg |
| CAS # | 1628208-23-0 |
| Pricing | 50 mg, USD $720.0 |
| Biological Activity | CPI-455 is a specific, pan-KDM5 inhibitor with an IC50 of 10 nM for KDM5A. CPI-455 mediates KDM5 inhibition, elevates global levels of H3K4me3, and decreases the number of drug-tolerant persister cancer cells in multiple cancer cell line models treated with standard chemotherapy or targeted agents[1]. |
| Purity | 98.95% |
| MWt | 278.31 |
| Formula | C₁₆H₁₄N₄O |