GW9508
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-15589-100 mg |
| CAS # | 885101-89-3 |
| Pricing | 100 mg, USD $290.0 |
| Biological Activity | GW9508 is a potent and selective G protein-coupled receptors FFA1 (GPR40) and GPR120 agonist with pEC50s of 7.32 and 5.46, respectively. GW9508 shows ~100-fold selectivity for GPR40 over GPR120. GW9508 is inactive against other GPCRs, kinases, proteases, integrins and PPARs. GW9508 is a glucose-sensitive insulin secretagogue and an ATP-sensitive potassium (KATP) channels opener. Anti-inflammatory and anti-atherosclerotic activities[1][2][3][4]. |
| Purity | 99.64% |
| MWt | 347.41 |
| Formula | C₂₂H₂₁NO₃ |