Umbralisib hydrochloride

Supplier MedChemExpress
Product # HY-12279C-100 mg
CAS # 1532533-78-0
Pricing 100 mg, USD $990.0
Synonyms TGR-1202 hydrochloride; RP5264 hydrochloride
MWt 608.01
Formula C₃₁H₂₅ClF₃N₅O₃
Biological Activity Umbralisib hydrochloride (TGR-1202 hydrochloride) is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM and 24.3 nM, respectively; Umbralisib hydrochloride (TGR-1202 hydrochloride) is also active against CK1ε, with an EC50 value of 6.0 μM.
Purity 99.63%
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