Umbralisib hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-12279C-100 mg |
| CAS # | 1532533-78-0 |
| Pricing | 100 mg, USD $990.0 |
| Synonyms | TGR-1202 hydrochloride; RP5264 hydrochloride |
| MWt | 608.01 |
| Formula | C₃₁H₂₅ClF₃N₅O₃ |
| Biological Activity | Umbralisib hydrochloride (TGR-1202 hydrochloride) is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM and 24.3 nM, respectively; Umbralisib hydrochloride (TGR-1202 hydrochloride) is also active against CK1ε, with an EC50 value of 6.0 μM. |
| Purity | 99.63% |