CRTh2 antagonist 3
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-135773 |
| CAS # | 312928-72-6 |
| Pricing | inquire |
| Biological Activity | CRTh2 antagonist 3 is a potent chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTh2) antagonist[1]. CRTh2 antagonist 3 enhances the activity of PDK1 toward a short peptide substrate, with an EC50 of 2 μM and a Kd of 8.4 μM. CRTh2 antagonist 3 has the potential for cardiovascular inflammation[2]. |
| MWt | 356.44 |
| Formula | C₁₉H₂₀N₂O₃S |