Quiflapon
Supplier | MedChemExpress |
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Product # | HY-10037-50 mg |
CAS # | 136668-42-3 |
Pricing | 50 mg, USD $931.0 |
Biological Activity | Quiflapon (MK-591) is a selective and specific 5-lipoxygenase-activating protein (FLAP) inhibitor with an IC50 of 1.6 nM in a FLAP binding assay. Quiflapon is also a potent and orally active Leukotriene biosynthesis (LT) inhibitor, shows IC50 values of 3.1 and 6.1 nM in intact human and elicited rat PMNLs, respectively. Quiflapon induces cell apoptosis[1][2]. |
Synonyms | MK-591 |
MWt | 587.17 |
Formula | C₃₄H₃₅ClN₂O₃S |