LP-922761
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-120179-100 mg |
| CAS # | 1454808-95-7 |
| Pricing | 100 mg, USD $1200.0 |
| Biological Activity | LP-922761 is a potent, selective and orally active adapter protein-2 associated kinase 1 (AAK1) inhibitor with IC50s of 4.8 nM and 7.6 nM in enzyme and cell assays, respectively. LP-922761 also inhibits BMP-2-inducible protein kinase (BIKE) with an IC50 of 24 nM. LP-922761 exhibits no significant activity at cyclin G-associated kinase (GAK), opioid, adrenergic α2 or GABAa receptors[1]. |
| Purity | 99.94% |
| MWt | 410.47 |
| Formula | C₂₁H₂₆N₆O₃ |