KDM2A/7A-IN-1

KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable histone lysine demethylases KDM2A/7A inhibitor, with an IC50 of 0.16 μM for KDM2A. It shows 75-fold selectivity over other JmjC lysine demethylases, and has no activity against methyltransferases and histone acetyltransferases.
Supplier BOC Sciences
Product # 2169272-46-0
Pricing Inquire
Cas 2169272-46-0
Molecular Weight 506.68
Molecular Formula C33H38N4O
Canonical SMILES CC(=O)N1C(C(C2=CC=CC=C21)(C#N)C3=CC=CC=C3)C4=CN=CC(=C4)CCCCCCCN5CCCC5
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