Cenerimod
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-17606-2 mg |
| CAS # | 1262414-04-9 |
| Pricing | 2 mg, USD $50.0 |
| Synonyms | ACT-334441 |
| MWt | 453.53 |
| Formula | C₂₅H₃₁N₃O₅ |
| Biological Activity | Cenerimod (ACT-334441) is a potent, selective and orally active S1P1 receptor modulator, with an EC50 of 1 nM. Cenerimod shows more than 36‐fold selctivity for hS1P1 over hS1P2, hS1P3, hS1P4, and hS1P5 receptor subtypes (EC50s=>10000, 228, 2134, and 36 nM, respectively). Cenerimod can attenuate murine experimental autoimmune encephalomyelitis (EAE) and murine sclerodermatous[1][2]. |
| Purity | ≥98.0% |