GSK2798745
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-19765-10 mg |
| CAS # | 1419609-94-1 |
| Pricing | 10 mg, USD $1250.0 |
| Biological Activity | GSK2798745 is a first-in-class, highly potent, selective, orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively. GSK2798745 is used in research for the treatment of pulmonary edema associated with congestive heart failure[1][2]. |
| Purity | 98.27% |
| MWt | 460.53 |
| Formula | C₂₅H₂₈N₆O₃ |