PD176252
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-103286-10 mM * 1 mL |
| CAS # | 204067-01-6 |
| Pricing | 10 mM * 1 mL, USD $90.0 |
| Biological Activity | PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; PD176252 is also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells. |
| Purity | ≥99.0% |
| MWt | 584.67 |
| Formula | C₃₂H₃₆N₆O₅ |