SCH442416
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-103169-10 mM * 1 mL |
| CAS # | 316173-57-6 |
| Pricing | 10 mM * 1 mL, USD $110.0 |
| Biological Activity | SCH442416 is a potent, selective and brain-penetrant antagonist of adenosine A2A receptor (A2AR), with Kis of 0.048 and 0.5 nM for human and rat A2AR respectively. SCH442416 displays more than 23000-fold selectivity over A1R, A2BR, and A3R (Ki=1111, 10000, and 10000 nM, respectively). SCH442416 can be used for imaging of adenosine A2A receptors in rat and primate brain[1][2]. |
| Purity | 98.19% |
| MWt | 389.41 |
| Formula | C₂₀H₁₉N₇O₂ |