BMS-986122
BMS-986122 is a selective, potent positive allosteric modulator of the mu-opioid receptor (µ-OR), shows potentiation of orthosteric agonist-mediated β-arrestin recruitment, adenylyl cyclase inhibition, and G protein activation, and potentiates DAMGO-mediated [35S]GTPγS binding in mouse brain membranes.
Supplier | Selleck Chemicals |
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Product # | E0472 |
Sku # | E0472-5mg |
Pricing | 5mg, $270.00 |