SB-657510
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-10656-5 mg |
| CAS # | 474960-44-6 |
| Pricing | 5 mg, USD $460.0 |
| Biological Activity | SB-657510 is a selective urotensin II (UII) receptor (UT) antagonist. The Ki values are 61, 17, 30, 65 and 56 nM for human, monkey, cat, rat and mouse receptors, respectively. SB-657510 exerts anti-inflammatory effects by inhibiting UII-induced upregulation of inflammatory mediators such as adhesion molecules, cytokines, and tissue factor in human vascular endothelial cells[1][2]. |
| Purity | 99.76% |
| MWt | 505.81 |
| Formula | C₁₉H₂₂BrClN₂O₅S |