CCG-50014
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-13509-10 mM * 1 mL |
| CAS # | 883050-24-6 |
| Pricing | 10 mM * 1 mL, USD $59.0 |
| Biological Activity | CCG-50014 is the most potent against the regulator of G-protein signaling protein type 4 (RGS4) (IC50 =30 nM) and is >20-fold selective for RGS4 over other RGS proteins. CCG-50014 binds covalently to the RGS, forming an adduct on two cysteine residues located in an allosteric regulatory site[1]. CCG50014, reduces nociceptive responses and enhances opioid-mediated analgesic effects in the mouse formalin test[2]. |
| Purity | ≥99.0% |
| MWt | 316.35 |
| Formula | C₁₆H₁₃FN₂O₂S |