BQ-123 TFA
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-12378A |
| Pricing | inquire |
| Biological Activity | BQ-123 TFA is a potent and selective endothelin A (ETA) receptor antagonist with an IC50 of 7.3 nM and a Ki of 25 nM. BQ-123 TFA inhibits endothelin-1-mediated proliferation of human pulmonary artery smooth muscle cells and lowers blood pressure in different rat models of hypertension[1][2][3]. |
| MWt | 724.72 |
| Formula | C₃₃H₄₃F₃N₆O₉ |