PLX51107
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-111422-10 mg |
| CAS # | 1627929-55-8 |
| Pricing | 10 mg, USD $250.0 |
| Biological Activity | PLX51107 is a potent and selective BET inhibitor, with Kds of 1.6, 2.1, 1.7, and 5 nM for BD1 and 5.9, 6.2, 6.1, and 120 nM for BD2 of BRD2, BRD3, BRD4, and BRDT, respectively; PLX51107 also interacts with the bromodomains of CBP and EP300 (Kd, in the 100 nM range). |
| Purity | 99.81% |
| MWt | 438.48 |
| Formula | C₂₆H₂₂N₄O₃ |