CNX-500
Supplier | MedChemExpress |
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Product # | HY-100338-5 mg |
CAS # | 1202758-21-1 |
Pricing | 5 mg, USD $3500.0 |
Biological Activity | CNX-500 is a probe consisting of a covalent Btk inhibitor (CC-292) chemically linked to biotin. CNX-500 retains inhibitory activity against Btk (IC50 of 0.5 nM) and the ability to form a covalent bond with Btk. CNX-500 has low inhibitory effects on kinase epidermal growth factor receptor, and upstream Src-family kinases including Syk and Lyn[1]. |
Purity | 99.19% |
MWt | 961.18 |
Formula | C₄₈H₆₈N₁₀O₉S |