FG 7142
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-100991-10 mg |
| CAS # | 78538-74-6 |
| Pricing | 10 mg, USD $200.0 |
| Synonyms | ZK 39106; LSU-65 |
| MWt | 225.25 |
| Formula | C₁₃H₁₁N₃O |
| Biological Activity | FG 7142 (ZK 39106; LSU-65), a non-selectively benzodiazepine inverse agonist, has high affinity for the α1 subunit-containing GABAA receptor (Ki=91 nM). FG 7142 (ZK 39106; LSU-65) also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 (ZK 39106; LSU-65) can increase tyrosine hydroxylation and cause upregulation of β-adrenoceptors in mouse cerebral cortex[1]. |
| Purity | ≥99.0% |