GKA50
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-15671-10 mM * 1 mL |
| CAS # | 851884-87-2 |
| Pricing | 10 mM * 1 mL, USD $562.0 |
| Biological Activity | GKA50 is a potent glucokinase activator (EC50=33 nM at 5 mM glucose). GKA50 stimulates insulin release from mouse islets of Langerhans. GKA50 is a glucose-like activator of beta-cell metabolism in rodent and human islets and a Ca2+-dependent modulator of insulin secretion. GKA50 shows significant glucose lowering in high fat fed female rats[1][2][3][4]. |
| Purity | ≥98.0% |
| MWt | 464.51 |
| Formula | C₂₆H₂₈N₂O₆ |