Talarozole
Supplier | MedChemExpress |
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Product # | HY-14531-5 mg |
CAS # | 201410-53-9 |
Pricing | 5 mg, USD $168.0 |
Synonyms | R115866 |
MWt | 377.51 |
Formula | C₂₁H₂₃N₅S |
Biological Activity | Talarozole (R115866) is an oral systemic all-trans retinoic acid metabolism blocking agent (RAMBA) which increases intracellular levels of endogenous all-trans retinoic acid (RA). Talarozole inhibits both CYP26A1 and CYP26B1 with IC50s of 5.4 and 0.46 nM, respectively. |
Purity | 99.78% |