Mavatrep
Supplier | MedChemExpress |
---|---|
Product # | HY-16935-10 mM * 1 mL |
CAS # | 956274-94-5 |
Pricing | 10 mM * 1 mL, USD $462.0 |
Synonyms | JNJ-39439335 |
MWt | 422.44 |
Formula | C₂₅H₂₁F₃N₂O |
Biological Activity | Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6. |
Purity | 99.85% |