FGTI-2734 mesylate
Supplier | MedChemExpress |
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Product # | HY-128350A-10 mg |
Pricing | 10 mg, USD $650.0 |
Biological Activity | FGTI-2734 mesylate is a RAS C-terminal mimetic dual farnesyl transferase (FT) and geranylgeranyl transferase-1 (GGT) inhibitor with IC50s of 250 nM and 520 nM for FT and GGT, respectively. FGTI-2734 mesylate can prevent membrane localization of KRAS, hence solving KRAS resistance problem and thwarting mutant KRAS patient-derived pancreatic tumors[1]. |
Purity | 98.73% |
MWt | 606.73 |
Formula | C₂₇H₃₅FN₆O₅S₂ |