Metergoline
Supplier | MedChemExpress |
---|---|
Product # | HY-B1033-100 mg |
CAS # | 17692-51-2 |
Pricing | 100 mg, USD $132.0 |
Biological Activity | Metergoline is a serotonin (5-HT) receptor and dopamine receptors antagonist, with pKis of 8.64, 8.75 and 8.75 for 5-HT2A, 5-HT2B and 5-HT2C, respectively. Metergoline is a high-affinity ligand for the h5-HT7 receptor, with a Ki of 16 nM. Metergoline is also a reversible neural Na+ channels inhibitor. Metergoline is commonly used for the research of seasonal affective disorder, prolactin hormone regulation[1][2][3]. |
Purity | 99.74% |
MWt | 403.52 |
Formula | C₂₅H₂₉N₃O₂ |