Isamoltane hemifumarate
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-19578B |
| CAS # | 874882-92-5 |
| Pricing | inquire |
| Biological Activity | Isamoltane hemifumarate is a selective antagonist of 5-HT1B receptor, with an IC50 of 39 nM for inhibits the binding of [125I]ICYP to 5-HT1B recognition sites in rat brain membranes. Isamoltane hemifumarate is also a β-adrenoceptor ligand, with an IC50 of 8.4 nM. Isamoltane hemifumarate shows anxiolytic activity[1]. |
| MWt | 332.4 |
| Formula | C₁₆H₂₂N₂O₂.₁/₂C₄H₄O₄ |