KPT-6566
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-123847-5 mg |
| CAS # | 881487-77-0 |
| Pricing | 5 mg, USD $360.0 |
| Biological Activity | KPT-6566, a potent prolyl isomerase PIN1 inhibitor, covalently binds to the catalytic site of PIN1, selectively inhibits and degrades PIN1. KPT-6566 shows an IC50 of 640 nM and a Ki of 625.2 nM for PIN1 PPIase domain. Anti-cancer activity[1]. |
| Purity | ≥98.0% |
| MWt | 443.54 |
| Formula | C₂₂H₂₁NO₅S₂ |