DCLK1-IN-1

Supplier MedChemExpress
Product # HY-135985-5 mg
CAS # 2222635-15-4
Pricing 5 mg, USD $450.0
Biological Activity DCLK1-IN-1 is a selective, oral bioavailability in vivo-compatible chemical probe of the doublecortin like kinase 1 (DCLK1 kinase) domain. DCLK1-IN-1 inhibits DCLK1 and DCLK2 kinases (IC50: DCLK1=9.5/57.2 nM and DCLK2=31/103 nM in binding and kinase assay, respectively). DCLK1-IN-1 shows low toxicity, and can investigate DCLK1 biology and establish its role in cancer, like DCLK1+ pancreatic ductal adenocarcinoma (PDAC)[1].
Purity 99.48%
MWt 527.54
Formula C₂₆H₂₈F₃N₇O₂
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