UCSF924
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-125751-10 mg |
| CAS # | 1434515-70-4 |
| Pricing | 10 mg, USD $500.0 |
| Biological Activity | UCSF924 is a potent and specific dopamine D4 receptor (DRD4) partial agonist with a EC50 of 4.2 nM. UCSF924 has a high-affinity with a Ki value of 3 nM for DRD4 and shows no measurable affinity for D2, D3 or the F261V/L328F D4 mutant. UCSF924 is a 7.4-fold bias toward arrestin over Gαi/o signaling, referenced to quinpirole[1]. |
| Purity | ≥98.0% |
| MWt | 322.4 |
| Formula | C₂₀H₂₂N₂O₂ |