TBK1/IKKε-IN-4
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-124652 |
| CAS # | 1381930-17-1 |
| Pricing | inquire |
| Biological Activity | TBK1/IKKε-IN-4 is a 6-aminopyrazolopyrimidine derivative and a potent, selective TBK1 and IKKε inhibitor with IC50 values of 13 nM and 59 nM, respectively. TBK1/IKKε-IN-4 shows 100- to 1000-fold less activity against other protein kinases including PDK1, PI3K family members and mTOR[1]. |
| MWt | 533.62 |
| Formula | C₂₈H₃₅N₇O₄ |