Isofistularin-3
Isofistularin-3 is a direct, DNA-competitive DNMT1 inhibitor, with an IC50 of 13.5 μM. Isofistularin-3, as a DNA demethylating agent, induces cell cycle arrest and sensitization to TRAIL in cancer cells. Isofistularin-3 can be used as an ADC cytotoxin.
Supplier | BOC Sciences |
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Product # | BADC-00845 |
Pricing | Inquire |
Molecular Weight | 1114.01 |
Molecular Formula | C31H30Br6N4O11 |