Isofistularin-3

Isofistularin-3 is a direct, DNA-competitive DNMT1 inhibitor, with an IC50 of 13.5 μM. Isofistularin-3, as a DNA demethylating agent, induces cell cycle arrest and sensitization to TRAIL in cancer cells. Isofistularin-3 can be used as an ADC cytotoxin.
Supplier BOC Sciences
Product # BADC-00845
Pricing Inquire
Molecular Weight 1114.01
Molecular Formula C31H30Br6N4O11
Feedback