Vofopitant dihydrochloride

Supplier MedChemExpress
Product # HY-12143-10 mM * 1 mL
CAS # 168266-51-1
Pricing 10 mM * 1 mL, USD $389.0
Synonyms GR 205171A
MWt 505.36
Formula C₂₁H₂₅Cl₂F₃N₆O
Biological Activity Vofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist, inhibits [3H]SP binding to the NK1 receptor with pKi values of 9.5 and 10.6 in rat and human membranes respectively, acts as a potential broad-spectrum anti-emetic agent[1].
Purity 99.11%
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