Vofopitant dihydrochloride
Supplier | MedChemExpress |
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Product # | HY-12143-10 mM * 1 mL |
CAS # | 168266-51-1 |
Pricing | 10 mM * 1 mL, USD $389.0 |
Synonyms | GR 205171A |
MWt | 505.36 |
Formula | C₂₁H₂₅Cl₂F₃N₆O |
Biological Activity | Vofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist, inhibits [3H]SP binding to the NK1 receptor with pKi values of 9.5 and 10.6 in rat and human membranes respectively, acts as a potential broad-spectrum anti-emetic agent[1]. |
Purity | 99.11% |