Pralsetinib (BLU-667)

Pralsetinib (BLU-667, CS 3009, Gavreto) is a highly potent and selective RET (c-RET) inhibitor with an IC50 of 0.4 nM for WT RET. It also demonstrates potent activity (IC50 0.4 nmol/L) against common oncogenic RET alterations, including RET (M918T).

• Supplier: Selleck Chemicals
• Product #: S8716
• Sku #: S8716-5mg