BI-749327
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-111925-10 mg |
| CAS # | 2361241-23-6 |
| Pricing | 10 mg, USD $550.0 |
| Biological Activity | BI-749327 is a potent, high selectivity and orally bioavailable TRPC6 antagonist, with IC50s of 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6, respectively. BI-749327 is 85-fold more selective for mouse TRPC6 than TRPC3 and 42-fold versus TRPC7[1]. |
| Purity | 99.53% |
| MWt | 442.43 |
| Formula | C₂₃H₂₁F₃N₄O₂ |